|
PKC Activator |
Year |
Title |
Web link |
|
8-octyl-benzolactam-V9 |
2006 |
Design and synthesis of 8-octyl-benzolactam-V9, a selective activator
for protein kinase C epsilon and eta |
http://www.ncbi.nlm.nih.gov/entrez/query.fcgi?cmd=Retrieve&db=PubMed&dopt=Citation&list_uids=16640328 |
|
Bryostatin 1 |
1996 |
Preclinical pharmacology of the natural product anticancer agent
bryostatin 1, an activator of protein kinase C |
http://www.ncbi.nlm.nih.gov/entrez/query.fcgi?cmd=Retrieve&db=PubMed&dopt=Citation&list_uids=8631017 |
|
Bryostatin 1 |
1997 |
Potentiation of ara-C-induced apoptosis by the protein kinase C
activator bryostatin 1 in human leukemia cells (HL-60) involves a
process dependent upon c-Myc |
http://www.ncbi.nlm.nih.gov/entrez/query.fcgi?cmd=Retrieve&db=PubMed&dopt=Citation&list_uids=9337072 |
|
Bryostatin 1 |
1999 |
Inhibition of protein kinase C activator-mediated induction of p21CIP1
and p27KIP1 by deoxycytidine analogs in human leukemia cells:
relationship to apoptosis and differentiation |
http://www.ncbi.nlm.nih.gov/entrez/query.fcgi?cmd=Retrieve&db=PubMed&dopt=Citation&list_uids=10403525 |
|
Chechum |
1989 |
Chechum (poison sap tree) toxin, a potent activator of protein kinase C |
http://www.ncbi.nlm.nih.gov/entrez/query.fcgi?cmd=Retrieve&db=PubMed&dopt=Citation&list_uids=2566840 |
|
Chloroform |
1987 |
Tumor promoter chloroform is a potent protein kinase C activator |
http://www.ncbi.nlm.nih.gov/entrez/query.fcgi?cmd=Retrieve&db=PubMed&dopt=Citation&list_uids=3827900 |
|
Cholesterol sulfate |
1994 |
Cholesterol sulfate, a novel activator for the eta isoform of protein
kinase C |
http://www.ncbi.nlm.nih.gov/entrez/query.fcgi?cmd=Retrieve&db=PubMed&dopt=Citation&list_uids=7819131 |
|
Daphnoretin |
1993 |
Daphnoretin, a new protein kinase C activator isolated from Wikstroemia
indica C.A. Mey |
http://www.ncbi.nlm.nih.gov/entrez/query.fcgi?cmd=Retrieve&db=PubMed&dopt=Citation&list_uids=8216237 |
|
Decursin |
1996 |
Decursin: a cytotoxic agent and protein kinase C activator from the root
of Angelica gigas |
http://www.ncbi.nlm.nih.gov/entrez/query.fcgi?cmd=Retrieve&db=PubMed&dopt=Citation&list_uids=8720379 |
|
Diazoxide |
2006 |
Diazoxide acts more as a PKC-epsilon activator, and indirectly activates
the mitochondrial K(ATP) channel conferring cardioprotection against
hypoxic injury |
http://www.ncbi.nlm.nih.gov/entrez/query.fcgi?cmd=Retrieve&db=PubMed&dopt=Citation&list_uids=17043673 |
|
DiC8 |
1997 |
Platelet activation with combination of ionophore A23187 and a direct
protein kinase C activator induces normal secretion in patients with
impaired receptor mediated secretion and abnormal signal transduction |
http://www.ncbi.nlm.nih.gov/entrez/query.fcgi?cmd=Retrieve&db=PubMed&dopt=Citation&list_uids=9526952 |
|
diC8 |
1999 |
In Hydra magnipapillata the activator of protein kinase C diC8 causes
multiple head formation along the body axis only when accompanied by
feeding, but heavy feeding alone is sufficient to cause multiple head
formation |
http://www.ncbi.nlm.nih.gov/entrez/query.fcgi?cmd=Retrieve&db=PubMed&dopt=Citation&list_uids=10707905 |
|
Farnesyl thiotriazole |
1995 |
Farnesyl thiotriazole, a potent neutrophil agonist and structurally
novel activator of protein kinase C |
http://www.ncbi.nlm.nih.gov/entrez/query.fcgi?cmd=Retrieve&db=PubMed&dopt=Citation&list_uids=7696255 |
|
Mezerein |
1994 |
Stimulation of calcium sequestration by mezerein, a protein kinase C
activator, in saponized rabbit platelets. |
http://www.ncbi.nlm.nih.gov/entrez/query.fcgi?cmd=Retrieve&db=PubMed&dopt=Citation&list_uids=7926583 |
|
Mezerein |
2001 |
Remyelination in vitro following protein kinase C activator-induced
demyelination |
http://www.ncbi.nlm.nih.gov/entrez/query.fcgi?cmd=Retrieve&db=PubMed&dopt=Citation&list_uids=11519722 |
|
PEP005 |
2005 |
PEP005, a selective small-molecule activator of protein kinase C, has
potent antileukemic activity mediated via the delta isoform of PKC |
http://www.ncbi.nlm.nih.gov/entrez/query.fcgi?cmd=Retrieve&db=PubMed&dopt=Citation&list_uids=15845901 |
|
psi(epsilon)RACK |
2003 |
Additive protection of the ischemic heart ex vivo by combined treatment
with delta-protein kinase C inhibitor and epsilon-protein kinase C
activator |
http://www.ncbi.nlm.nih.gov/entrez/query.fcgi?cmd=Retrieve&db=PubMed&dopt=Citation&list_uids=12860903 |
|
Sapintoxin A |
1987 |
Sapintoxin A. A fluorescent phorbol ester that is a potent activator of
protein kinase C but is not a tumour promoter |
http://www.ncbi.nlm.nih.gov/entrez/query.fcgi?cmd=Retrieve&db=PubMed&dopt=Citation&list_uids=3690506 |
|
TPA |
1992 |
Activation of protein kinase C increases phosphorylation of the L-myc
trans-activator domain at a GSK-3 target site |
http://www.ncbi.nlm.nih.gov/entrez/query.fcgi?cmd=Retrieve&db=PubMed&dopt=Citation&list_uids=1312697 |
